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CRYSTAL STRUCTURE OF BRUTON'S TYROSINE KINASE IN COMPLEX WITH INHIBITOR CGI2625

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Protein Data Bank Japan2023-10-04 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6aua
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CRYSTAL STRUCTURE OF BRUTON'S TYROSINE KINASE IN COMPLEX WITH INHIBITOR CGI2625 Descriptor: GLYCEROL, N-{3-[(2R)-6-{[3-amino-4-(morpholine-4-carbonyl)phenyl]amino}-5-oxo-2,5-dihydropyrazin-2-yl]-2-methylphenyl}-4-(piperidin-1-yl)benzamide, SULFATE ION, ... Authors: Davies, D.R, Staker, B.L. Deposit date: 2017-08-31 Release date: 2018-09-12 Last modified: 2023-10-04 Method: X-RAY DIFFRACTION (1.66 Å) Cite: To Be Determined TO BE PUBLISHED

布鲁顿酪氨酸激酶(Bruton's Tyrosine Kinase)与抑制剂CGI2625复合物的晶体结构 描述符:甘油、N-{3-[(2R)-6-{[3-氨基-4-(吗啉-4-羰基)苯基]氨基}-5-氧代-2,5-二氢吡嗪-2-基]-2-甲基苯基}-4-(哌啶-1-基)苯甲酰胺、硫酸根离子,…… 作者:Davies, D.R.、Staker, B.L. 提交日期:2017-08-31 发布日期:2018-09-12 最后修改日期:2023-10-04 检测方法:X射线衍射(X-RAY DIFFRACTION),分辨率1.66埃(Å) 引用信息:待确定,即将发表
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2017-08-31
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