Toxoplasma gondii Enoyl acyl carrier protein reductase
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Toxoplasma gondii Enoyl acyl carrier protein reductase Descriptor: Enoyl-acyl carrier reductase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE Authors: Muench, S.P, Wilkinson, C, Prigge, S.T, Rice, D.W. Deposit date: 2013-12-16 Release date: 2014-02-05 Last modified: 2024-04-03 Method: X-RAY DIFFRACTION (2 Å) Cite: The benzimidazole based drugs show good activity against T. gondii but poor activity against its proposed enoyl reductase enzyme target Bioorg.Med.Chem.Lett., 24, 2014
刚地弓形虫(Toxoplasma gondii)烯酰酰基载体蛋白还原酶(Enoyl acyl carrier protein reductase)
描述:烯酰-酰基载体蛋白还原酶(Enoyl-acyl carrier reductase),烟酰胺腺嘌呤二核苷酸(NICOTINAMIDE-ADENINE-DINUCLEOTIDE)
作者:Muench, S.P.、Wilkinson, C.、Prigge, S.T.、Rice, D.W.
提交日期:2013-12-16
发布日期:2014-02-05
最后修改日期:2024-04-03
方法:X射线衍射(X-RAY DIFFRACTION),分辨率2埃(2 Å)
引用:苯并咪唑类药物对刚地弓形虫表现出良好活性,但对其推定的烯酰还原酶靶标酶活性较差,《Bioorg.Med.Chem.Lett.》,24,2014
创建时间:
2013-12-16



