Crystal structure of mutant AR-LBD (Y764C) bound to dihydrotestosterone
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Crystal structure of mutant AR-LBD (Y764C) bound to dihydrotestosterone Descriptor: 5-ALPHA-DIHYDROTESTOSTERONE, Androgen receptor, IMIDAZOLE, ... Authors: Alegre-Marti, A, Jimenez-Panizo, A, Estebanez-Perpina, E, Fuentes-Prior, P. Deposit date: 2022-05-11 Release date: 2023-03-22 Last modified: 2024-02-07 Method: X-RAY DIFFRACTION (1.4 Å) Cite: A hotspot for posttranslational modifications on the androgen receptor dimer interface drives pathology and anti-androgen resistance. Sci Adv, 9, 2023
与二氢睾酮结合的Y764C突变型雄激素受体配体结合域(Androgen Receptor Ligand Binding Domain, AR-LBD)晶体结构
描述符:5-α-二氢睾酮、雄激素受体、咪唑(IMIDAZOLE)等
作者:Alegre-Marti, A、Jimenez-Panizo, A、Estebanez-Perpina, E、Fuentes-Prior, P
沉积日期:2022-05-11
发布日期:2023-03-22
最后修改日期:2024-02-07
实验方法:X射线衍射(1.4埃)
引用文献:《雄激素受体二聚体界面的翻译后修饰热点驱动病理发生与抗雄激素耐药性》,发表于《科学进展》(Science Advances),2023年,第9卷
创建时间:
2022-05-11



