Crystal Structure of Human Chymase in Complex with Fragment Inhibitor 6-chloro-2,3-dihydro-1H-isoindol-1-one
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Crystal Structure of Human Chymase in Complex with Fragment Inhibitor 6-chloro-2,3-dihydro-1H-isoindol-1-one Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 6-chloro-2,3-dihydro-1H-isoindol-1-one, Chymase, ... Authors: Collins, B.K, Padyana, A.K. Deposit date: 2013-04-15 Release date: 2013-05-29 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (1.8 Å) Cite: Discovery of Potent, Selective Chymase Inhibitors via Fragment Linking Strategies. J.Med.Chem., 56, 2013
人糜酶(Human Chymase)与片段抑制剂6-氯-2,3-二氢-1H-异吲哚-1-酮(6-chloro-2,3-dihydro-1H-isoindol-1-one)复合物的晶体结构
描述项:2-乙酰氨基-2-脱氧-β-D-吡喃葡萄糖(2-acetamido-2-deoxy-beta-D-glucopyranose)、6-氯-2,3-二氢-1H-异吲哚-1-酮、糜酶(Chymase)……
作者:Collins, B.K, Padyana, A.K.
提交日期:2013-04-15
发布日期:2013-05-29
最后修改日期:2024-11-20
实验方法:X射线衍射(1.8 Å)
引用文献:Discovery of Potent, Selective Chymase Inhibitors via Fragment Linking Strategies. J.Med.Chem., 56, 2013
创建时间:
2013-04-15



