Cryogenic Human Hsp90a-NTD bound to EC144
收藏Protein Data Bank Japan2023-10-18 更新2026-04-19 收录
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Cryogenic Human Hsp90a-NTD bound to EC144 Descriptor: 5-{2-amino-4-chloro-7-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-7H-pyrrolo[2,3-d]pyrimidin-5-yl}-2-methylpent-4-yn-2 -ol, Heat shock protein HSP 90-alpha, MAGNESIUM ION Authors: Stachowski, T.R, Vanarotti, M, Seetharaman, J, Fischer, M. Deposit date: 2021-09-21 Release date: 2022-08-03 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.45 Å) Cite: Water Networks Repopulate Protein-Ligand Interfaces with Temperature. Angew.Chem.Int.Ed.Engl., 61, 2022
结合EC144的低温冷冻人类热休克蛋白90α N端结构域(Hsp90α-NTD)
配体描述:5-{2-氨基-4-氯-7-[(4-甲氧基-3,5-二甲基吡啶-2-基)甲基]-7H-吡咯并[2,3-d]嘧啶-5-基}-2-甲基戊-4-炔-2-醇
蛋白组分:热休克蛋白HSP 90-α、镁离子
作者:Stachowski T.R.、Vanarotti M.、Seetharaman J.、Fischer M.
存入日期:2021-09-21
发布日期:2022-08-03
最后修改日期:2023-10-18
实验方法:X射线衍射(1.45 Å)
引用文献:《Water Networks Repopulate Protein-Ligand Interfaces with Temperature》,《Angew.Chem.Int.Ed.Engl.》,第61卷,2022年
创建时间:
2021-09-21



