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Human CDK8/Cyclin-C complex with inhibitor 2-9

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Protein Data Bank Japan2025-02-05 更新2026-04-19 收录
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Human CDK8/Cyclin-C complex with inhibitor 2-9 Descriptor: 1,2-ETHANEDIOL, 4-[(3~{S})-3-[2-[(3~{R})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]piperidin-1-yl]carbonyl-1~{H}-pyrrole-2-carbonitrile, Cyclin-C, ... Authors: Somers, D.O. Deposit date: 2024-10-29 Release date: 2025-01-22 Last modified: 2025-02-05 Method: X-RAY DIFFRACTION (2.573 Å) Cite: Phenotype-Led Identification of IL-10 Upregulators in Human CD4 + T-cells and Elucidation of Their Pharmacology as Highly Selective CDK8/CDK19 Inhibitors. J.Med.Chem., 68, 2025
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2024-10-29
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