Caspase 3 Bound to a covalent inhibitor
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Caspase 3 Bound to a covalent inhibitor Descriptor: (3S)-3-({[(5S,10aS)-2-{(2S)-4-carboxy-2-[(phenylacetyl)amino]butyl}-1,3-dioxo-2,3,5,7,8,9,10,10a-octahydro-1H-[1,2,4]triazolo[1,2-a]cinnolin-5-yl]carbonyl}amino)-4-oxopentanoic acid, Caspase-3 Authors: Kamtekar, S, Watt, W, Finzel, B.C, Harris, M.S, Blinn, J, Wang, Z, Tomasselli, A.G. Deposit date: 2009-11-03 Release date: 2010-08-11 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2 Å) Cite: Kinetic and structural characterization of caspase-3 and caspase-8 inhibition by a novel class of irreversible inhibitors. Biochim.Biophys.Acta, 1804, 2010
创建时间:
2009-11-03



