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Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor H10

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor H10 Descriptor: 3-[2-[4-[2-[[4-[(3-aminocarbonylphenyl)amino]-4-oxidanylidene-butanoyl]amino]ethyl]-1,2,3-triazol-1-yl]ethylsulfamoyl]benzoic acid, Poly [ADP-ribose] polymerase 14 Authors: Karlberg, T, Thorsell, A.G, Schuler, H. Deposit date: 2016-09-28 Release date: 2016-12-21 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.17 Å) Cite: Small Molecule Microarray Based Discovery of PARP14 Inhibitors. Angew. Chem. Int. Ed. Engl., 56, 2017
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2016-09-28
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