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JAK2 kinase (JH1 domain) mutant P1057A in complex with TG101209

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5hez
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资源简介:
JAK2 kinase (JH1 domain) mutant P1057A in complex with TG101209 Descriptor: CHLORIDE ION, N-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamide, Tyrosine-protein kinase JAK2, ... Authors: Ultsch, M, Eigenbrot, C. Deposit date: 2016-01-06 Release date: 2016-11-09 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.66 Å) Cite: Resolving TYK2 locus genotype-to-phenotype differences in autoimmunity. Sci Transl Med, 8, 2016
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2016-01-06
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