CDK2/cyclin A2 in complex with pyrazolo[4,3-d]pyrimidine inhibitor LGR4455
收藏Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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CDK2/cyclin A2 in complex with pyrazolo[4,3-d]pyrimidine inhibitor LGR4455 Descriptor: 1,2-ETHANEDIOL, 5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{N}-[(4-pyridin-2-ylphenyl)methyl]-2~{H}-pyrazolo[4,3-d]pyrimidin-7-amine, BROMIDE ION, ... Authors: Skerlova, J, Rezacova, P. Deposit date: 2018-06-20 Release date: 2019-05-01 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.15 Å) Cite: 3,5,7-Substituted Pyrazolo[4,3- d]pyrimidine Inhibitors of Cyclin-Dependent Kinases and Their Evaluation in Lymphoma Models. J.Med.Chem., 62, 2019
创建时间:
2018-06-20



