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Protein kinase Pim-1 in complex with small molecule inibitor

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Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2xj1
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Protein kinase Pim-1 in complex with small molecule inibitor Descriptor: (2E)-3-(3-{6-[(TRANS-4-AMINOCYCLOHEXYL)AMINO]PYRAZIN-2-YL}PHENYL)PROP-2-ENOIC ACID, PROTO-ONCOGENE SERINE/THREONINE-PROTEIN KINASE PIM-1 Authors: Schulz, M.N, Fanghanel, J, Schafer, M, Badock, V, Briem, H, Boemer, U, Nguyen, D, Husemann, M, Hillig, R.C. Deposit date: 2010-07-01 Release date: 2011-02-23 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.13 Å) Cite: Crystallographic Fragment Screen Identifies Cinnamic Acid Derivatives as Starting Points for Potent Pim-1 Inhibitors Acta Crystallogr.,Sect.D, 67, 2011
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2010-07-01
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