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Human PPARgamma ligand-binding domain R288A mutant in complex with imatinib

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Protein Data Bank Japan2023-11-22 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6ktn
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资源简介:
Human PPARgamma ligand-binding domain R288A mutant in complex with imatinib Descriptor: 16-mer peptide from Nuclear receptor coactivator 1, 4-(4-METHYL-PIPERAZIN-1-YLMETHYL)-N-[4-METHYL-3-(4-PYRIDIN-3-YL-PYRIMIDIN-2-YLAMINO)-PHENYL]-BENZAMIDE, Peroxisome proliferator-activated receptor gamma Authors: Jang, J.Y, Han, B.W. Deposit date: 2019-08-28 Release date: 2020-02-05 Last modified: 2023-11-22 Method: X-RAY DIFFRACTION (2.752 Å) Cite: Structural Basis for the Regulation of PPAR gamma Activity by Imatinib. Molecules, 24, 2019
创建时间:
2019-08-28
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