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Crystal structure of GSK-3 beta in complex with NMS-869553A

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Protein Data Bank Japan2023-08-30 更新2026-03-21 收录
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Crystal structure of GSK-3 beta in complex with NMS-869553A Descriptor: (7S)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-one, Glycogen synthase kinase-3 beta Authors: Bossi, R.T. Deposit date: 2008-07-17 Release date: 2009-03-03 Last modified: 2023-08-30 Method: X-RAY DIFFRACTION (2.2 Å) Cite: First Cdc7 kinase inhibitors: pyrrolopyridinones as potent and orally active antitumor agents. 2. Lead discovery. J.Med.Chem., 52, 2009
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2008-07-17
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