Crystal structure of the first bromodomain of human BRD4 in complex with SJ001010551-2
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Crystal structure of the first bromodomain of human BRD4 in complex with SJ001010551-2 Descriptor: 1,2-ETHANEDIOL, 2-[(6S,10S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]-N-[(pyridin-2-yl)methyl]acetamide, Bromodomain-containing protein 4 Authors: Stachowski, T.R, Fischer, M. Deposit date: 2021-07-28 Release date: 2022-08-03 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.05 Å) Cite: From PROTAC to inhibitor: Structure-guided discovery of potent and orally bioavailable BET inhibitors. Eur.J.Med.Chem., 251, 2023
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2021-07-28
