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Joint X-ray/neutron structure of HIV-1 protease triple mutant (V32I,I47V,V82I) with amprenavir at pH 6.0

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Protein Data Bank Japan2024-04-03 更新2026-03-21 收录
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Joint X-ray/neutron structure of HIV-1 protease triple mutant (V32I,I47V,V82I) with amprenavir at pH 6.0 Descriptor: Protease, {3-[(4-AMINO-BENZENESULFONYL)-ISOBUTYL-AMINO]-1-BENZYL-2-HYDROXY-PROPYL}-CARBAMIC ACID TETRAHYDRO-FURAN-3-YL ESTER Authors: Kovalevsky, A.Y, Gerlits, O.O. Deposit date: 2016-09-07 Release date: 2017-03-01 Last modified: 2024-04-03 Method: NEUTRON DIFFRACTION (1.85 Å), X-RAY DIFFRACTION Cite: Room Temperature Neutron Crystallography of Drug Resistant HIV-1 Protease Uncovers Limitations of X-ray Structural Analysis at 100 K. J. Med. Chem., 60, 2017
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2016-09-07
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