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Aurora-A in complex with shape-diverse fragment 39

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Protein Data Bank Japan2024-11-20 更新2026-03-21 收录
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Aurora-A in complex with shape-diverse fragment 39 Descriptor: (1~{S},10~{S})-12-cyclopropyl-1-oxidanyl-10-propan-2-yl-9,12-diazatricyclo[8.2.1.0^{2,7}]trideca-2(7),3,5-trien-11-one, ADENOSINE-5'-DIPHOSPHATE, Aurora kinase A, ... Authors: Bayliss, R, McIntyre, P.J. Deposit date: 2019-03-22 Release date: 2019-05-08 Last modified: 2024-11-20 Method: X-RAY DIFFRACTION (2.209 Å) Cite: Construction of a Shape-Diverse Fragment Set: Design, Synthesis and Screen against Aurora-A Kinase. Chemistry, 25, 2019

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2019-03-22
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