Human Brd2(BD2) mutant in complex with ME
收藏Protein Data Bank Japan2024-01-17 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5o39
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Human Brd2(BD2) mutant in complex with ME Descriptor: (2~{S})-1-[(2~{S})-2-oxidanylpropoxy]propan-2-ol, Bromodomain-containing protein 2, CHLORIDE ION, ... Authors: Runcie, A.C, Chan, K.-H, Ciulli, A. Deposit date: 2017-05-23 Release date: 2018-02-14 Last modified: 2024-01-17 Method: X-RAY DIFFRACTION (1.74 Å) Cite: Optimization of a "bump-and-hole" approach to allele-selective BET bromodomain inhibition. Chem Sci, 9, 2018
创建时间:
2017-05-23



