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Discovery of novel, orally efficacious Liver X Receptor (LXR) beta agonists

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Protein Data Bank Japan2023-09-27 更新2026-03-21 收录
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Discovery of novel, orally efficacious Liver X Receptor (LXR) beta agonists Descriptor: Oxysterols receptor LXR-beta,Nuclear receptor coactivator 2, Retinoic acid receptor RXR-beta,Nuclear receptor coactivator 2, {2-[(2R)-4-[4-(hydroxymethyl)-3-(methylsulfonyl)phenyl]-2-(propan-2-yl)piperazin-1-yl]-4-(trifluoromethyl)pyrimidin-5-yl}methanol Authors: Chen, G, McKeever, B.M. Deposit date: 2016-02-12 Release date: 2016-06-29 Last modified: 2023-09-27 Method: X-RAY DIFFRACTION (2.61 Å) Cite: Discovery of a Novel, Orally Efficacious Liver X Receptor (LXR) beta Agonist. J.Med.Chem., 59, 2016
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2016-02-12
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