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Crystal structure of the first bromodomain (BD1) of human BRD3 bound to ERK5-IN-1

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Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Crystal structure of the first bromodomain (BD1) of human BRD3 bound to ERK5-IN-1 Descriptor: 11-cyclopentyl-2-({2-ethoxy-4-[4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]phenyl}amino)-5-methyl-5,11-dihydro-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one, Bromodomain-containing protein 3 Authors: Karim, M.R, Bikowitz, M.J, Schonbrunn, E. Deposit date: 2021-01-07 Release date: 2021-07-14 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (2.302 Å) Cite: Differential BET Bromodomain Inhibition by Dihydropteridinone and Pyrimidodiazepinone Kinase Inhibitors. J.Med.Chem., 64, 2021
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2021-01-07
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