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Structure of cytochrome P450 EryK cocrystallized with inhibitor clotrimazole.

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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Structure of cytochrome P450 EryK cocrystallized with inhibitor clotrimazole. Descriptor: 1-[(2-CHLOROPHENYL)(DIPHENYL)METHYL]-1H-IMIDAZOLE, DIMETHYL SULFOXIDE, ERYTHROMYCIN B/D C-12 HYDROXYLASE, ... Authors: Savino, C, Montemiglio, L.C, Gianni, S, Vallone, B. Deposit date: 2010-05-24 Release date: 2010-09-29 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (1.9 Å) Cite: Azole Drugs Trap Cytochrome P450 Eryk in Alternative Conformational States. Biochemistry, 49, 2010
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2010-05-24
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