five

Kinase domain of cSrc in complex with RL236

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Kinase domain of cSrc in complex with RL236 Descriptor: N-[4-({4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl}oxy)phenyl]prop-2-enamide, Proto-oncogene tyrosine-protein kinase Src Authors: Becker, C, Mayer-Wrangowski, S.C, Julian, E, Rauh, D. Deposit date: 2015-08-03 Release date: 2015-09-02 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.7 Å) Cite: Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach. J.Med.Chem., 58, 2015
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2015-08-03
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