IRAK4 IN COMPLEX WITH inhibitor
收藏Protein Data Bank Japan2024-10-23 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/6ti8
下载链接
链接失效反馈官方服务:
资源简介:
IRAK4 IN COMPLEX WITH inhibitor Descriptor: Interleukin-1 receptor-associated kinase 4, ~{N},~{N}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamide Authors: Xue, Y, Aagaard, A, Degorce, S.L. Deposit date: 2019-11-22 Release date: 2020-10-28 Last modified: 2024-10-23 Method: X-RAY DIFFRACTION (2.32 Å) Cite: Improving metabolic stability and removing aldehyde oxidase liability in a 5-azaquinazoline series of IRAK4 inhibitors. Bioorg.Med.Chem., 28, 2020
创建时间:
2019-11-22



