five

Crystal structure of PPARgamma ligand-binding domain in complex with ZINC5672437

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Protein Data Bank Japan2025-04-30 更新2026-04-19 收录
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Crystal structure of PPARgamma ligand-binding domain in complex with ZINC5672437 Descriptor: N-(4-carbamoylphenyl)-2-chloro-5-nitrobenzamide, Peroxisome proliferator-activated receptor gamma, nonanoic acid Authors: Shang, J, Kojetin, D.J. Deposit date: 2022-12-14 Release date: 2024-03-20 Last modified: 2025-04-30 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Ligand efficacy shifts a nuclear receptor conformational ensemble between transcriptionally active and repressive states. Nat Commun, 16, 2025
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2022-12-14
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