Crystal structure of PPARgamma ligand-binding domain in complex with ZINC5672437
收藏Protein Data Bank Japan2025-04-30 更新2026-04-19 收录
下载链接:
https://pdbj.org/mine/summary/8fhf
下载链接
链接失效反馈官方服务:
资源简介:
Crystal structure of PPARgamma ligand-binding domain in complex with ZINC5672437 Descriptor: N-(4-carbamoylphenyl)-2-chloro-5-nitrobenzamide, Peroxisome proliferator-activated receptor gamma, nonanoic acid Authors: Shang, J, Kojetin, D.J. Deposit date: 2022-12-14 Release date: 2024-03-20 Last modified: 2025-04-30 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Ligand efficacy shifts a nuclear receptor conformational ensemble between transcriptionally active and repressive states. Nat Commun, 16, 2025
创建时间:
2022-12-14



