Human tankyrase 2 - catalytic Parp domain in complex with an inhibitor UPF1854
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Human tankyrase 2 - catalytic Parp domain in complex with an inhibitor UPF1854 Descriptor: 4-{2-[(6-methyl[1,2,4]triazolo[4,3-b]pyridazin-8-yl)amino]ethyl}phenol, SULFATE ION, Tankyrase-2, ... Authors: Karlberg, T, Camaioni, E, Schuler, H. Deposit date: 2013-08-12 Release date: 2014-03-12 Last modified: 2023-09-20 Method: X-RAY DIFFRACTION (1.95 Å) Cite: Design, Synthesis, Crystallographic Studies, and Preliminary Biological Appraisal of New Substituted Triazolo[4,3-b]pyridazin-8-amine Derivatives as Tankyrase Inhibitors. J.Med.Chem., 57, 2014
创建时间:
2013-08-12



