P38ALPHA MAP KINASE BOUND TO CMPD 8
收藏Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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https://pdbj.org/mine/summary/4a9y
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P38ALPHA MAP KINASE BOUND TO CMPD 8 Descriptor: MITOGEN-ACTIVATED PROTEIN KINASE 14, N-(3-{[7-METHOXY-6-(2-PYRROLIDIN-1-YLETHOXY)QUINAZOLIN-4-YL]AMINO}-4-METHYLPHENYL)-2-MORPHOLIN-4-YLISONICOTINAMIDE Authors: Gerhardt, S, Hargreaves, D. Deposit date: 2011-11-29 Release date: 2012-05-16 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.2 Å) Cite: The Discovery of N-Cyclopropyl-4-Methyl-3-[6--(4-Methylpiperazin-1-Yl-4-Oxoquinazolin-3(4H)-Yl]Benzamide (Azd6703), a Clinical P38Alpha Map Kinase Inhibitor for the Treatment of Inflammatory Diseases Bioorg.Med.Chem.Lett., 22, 2012
创建时间:
2011-11-29



