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Crystal Structure of EGFR(L858R/T790M/C797S) in complex with Osimertinib

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Protein Data Bank Japan2023-11-29 更新2026-03-21 收录
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https://pdbj.org/mine/summary/6lud
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Crystal Structure of EGFR(L858R/T790M/C797S) in complex with Osimertinib Descriptor: Epidermal growth factor receptor, N-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1H-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide Authors: Kawauchi, H, Fukami, T.A, Sato, S, Endo, M, Torizawa, T, Kashima, K, Chiba, T, Sakamoto, H. Deposit date: 2020-01-27 Release date: 2020-10-07 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (2.05 Å) Cite: CH7233163 Overcomes Osimertinib-Resistant EGFR-Del19/T790M/C797S Mutation. Mol.Cancer Ther., 19, 2020
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2020-01-27
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