First bromodomain of BRD4 bound to inhibitor XD42
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First bromodomain of BRD4 bound to inhibitor XD42 Descriptor: 4-acetyl-N-[3-(azepan-1-ylsulfonyl)phenyl]-5-methyl-3-propyl-1H-pyrrole-2-carboxamide, Bromodomain-containing protein 4 Authors: Wohlwend, D, Huegle, M. Deposit date: 2015-08-06 Release date: 2016-01-20 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.2 Å) Cite: 4-Acyl Pyrrole Derivatives Yield Novel Vectors for Designing Inhibitors of the Acetyl-Lysine Recognition Site of BRD4(1). J.Med.Chem., 59, 2016
创建时间:
2015-08-06



