mPI3Kd IN COMPLEX WITH 7k
收藏Protein Data Bank Japan2024-05-08 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5t2i
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mPI3Kd IN COMPLEX WITH 7k Descriptor: 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-4-carboxamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform Authors: Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L. Deposit date: 2016-08-23 Release date: 2017-04-19 Last modified: 2024-05-08 Method: X-RAY DIFFRACTION (2.3 Å) Cite: Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
创建时间:
2016-08-23



