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Crystal structure of human KAT II-inhibitor complex

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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Crystal structure of human KAT II-inhibitor complex Descriptor: (3S)-10-(4-AMINOPIPERAZIN-1-YL)-9-FLUORO-7-HYDROXY-3-METHYL-2,3-DIHYDRO-8H-[1,4]OXAZINO[2,3,4-IJ]QUINOLINE-6-CARBOXYLATE, GLYCEROL, IODIDE ION, ... Authors: Rossi, F, Casazza, V, Garavaglia, S, Sathyasaikumar, K.V, Schwarcz, R, Kojima, S.I, Okuwaki, K, Ono, S.I, Kajii, Y, Rizzi, M. Deposit date: 2010-06-08 Release date: 2010-07-28 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.1 Å) Cite: Crystal Structure-Based Selective Targeting of the Pyridoxal 5'-Phsosphate Dependent Enzyme Kynurenine Aminotransferase II for Cognitive Enhancement J.Med.Chem., 53, 2010
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2010-06-08
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