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Trypanosoma brucei PTR1 in complex with inhibitor WHF30

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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https://pdbj.org/mine/summary/2yhu
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Trypanosoma brucei PTR1 in complex with inhibitor WHF30 Descriptor: 3-(5-AMINO-1,3,4-THIADIAZOL-2-YL)-1-THIOPHEN-2-YLPROPAN-1-ONE, ACETATE ION, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... Authors: Nerini, E, Dawson, A, Hunter, W.N, Costi, M.P. Deposit date: 2011-05-06 Release date: 2012-05-23 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (2.01 Å) Cite: Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To Inhibit Trypanosoma brucei Pteridine Reductase in Support of Early-Stage Drug Discovery. ACS Omega, 2, 2017
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2011-05-06
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