five

PDE10 complexed with 4,6-dichloro-2-cyclopropyl-5-methyl-pyrimidine

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Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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PDE10 complexed with 4,6-dichloro-2-cyclopropyl-5-methyl-pyrimidine Descriptor: 4,6-dichloro-2-cyclopropyl-5-methylpyrimidine, MAGNESIUM ION, ZINC ION, ... Authors: Yan, Y. Deposit date: 2015-06-15 Release date: 2015-09-30 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (1.7 Å) Cite: Discovery and Optimization of a Series of Pyrimidine-Based Phosphodiesterase 10A (PDE10A) Inhibitors through Fragment Screening, Structure-Based Design, and Parallel Synthesis. J.Med.Chem., 58, 2015
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2015-06-15
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