JAK3 with covalent inhibitor PF-06651600
收藏Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5toz
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JAK3 with covalent inhibitor PF-06651600 Descriptor: 1-{(2S,5R)-2-methyl-5-[(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}propan-1-one, SULFATE ION, Tyrosine-protein kinase JAK3 Authors: Vajdos, F.F. Deposit date: 2016-10-19 Release date: 2016-11-09 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (1.98 Å) Cite: Discovery of a JAK3-Selective Inhibitor: Functional Differentiation of JAK3-Selective Inhibition over pan-JAK or JAK1-Selective Inhibition. ACS Chem. Biol., 11, 2016
创建时间:
2016-10-19



