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Crystal structure of human choline alpha in complex with an inhibitor

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Protein Data Bank Japan2024-01-31 更新2026-03-21 收录
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Crystal structure of human choline alpha in complex with an inhibitor Descriptor: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 4-(6-azanyl-2-chloranyl-purin-9-yl)-~{N}-(4-methyl-1,3-thiazol-2-yl)cyclohexane-1-carboxamide, Choline kinase alpha, ... Authors: Casale, E, Fasolini, M. Deposit date: 2021-01-25 Release date: 2021-10-13 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Identification of unprecedented ATP-competitive choline kinase inhibitors. Bioorg.Med.Chem.Lett., 51, 2021
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2021-01-25
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