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Discovery and Pharmacological Characterization of Novel Quinazoline-based PI3K delta-selective Inhibitors

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Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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Discovery and Pharmacological Characterization of Novel Quinazoline-based PI3K delta-selective Inhibitors Descriptor: 5-{4-[3-(4-acetylpiperazine-1-carbonyl)phenyl]quinazolin-6-yl}-2-methoxypyridine-3-carbonitrile, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform Authors: Gutmann, S, Rummel, G, Shrestha, B. Deposit date: 2016-03-15 Release date: 2016-08-10 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.85 Å) Cite: Discovery and Pharmacological Characterization of Novel Quinazoline-Based PI3K Delta-Selective Inhibitors. Acs Med.Chem.Lett., 7, 2016
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2016-03-15
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