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Structure-based drug design of novel ASK1 inhibitors using a fully integrated lead optimization strategy

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Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
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Structure-based drug design of novel ASK1 inhibitors using a fully integrated lead optimization strategy Descriptor: Mitogen-activated protein kinase kinase kinase 5, N-(1-ethyl-1H-pyrazol-4-yl)furan-3-carboxamide Authors: Dougan, D.R, Lawson, J.D, Lane, W. Deposit date: 2017-03-01 Release date: 2017-03-29 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (3.1 Å) Cite: Structure-based drug design of novel ASK1 inhibitors using an integrated lead optimization strategy. Bioorg. Med. Chem. Lett., 27, 2017

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2017-03-01
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