Crystal structure of an Estrogen Receptor alpha 8-mer phosphopeptide in complex with 14-3-3sigma stabilized by Pyrrolidone1
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Crystal structure of an Estrogen Receptor alpha 8-mer phosphopeptide in complex with 14-3-3sigma stabilized by Pyrrolidone1 Descriptor: 14-3-3 protein sigma, 5-[(2R)-3-benzoyl-4-hydroxy-2-(4-nitrophenyl)-5-oxo-2,5-dihydro-1H-pyrrol-1-yl]-2-hydroxybenzoic acid, C-terminal phosphopeptide of human estrogen receptor alpha, ... Authors: Andrei, S.A, Bosica, F, Ottmann, C, O'Mahony, G. Deposit date: 2019-11-26 Release date: 2020-04-29 Last modified: 2026-04-15 Method: X-RAY DIFFRACTION (1.85 Å) Cite: Design of Drug-Like Protein-Protein Interaction Stabilizers Guided By Chelation-Controlled Bioactive Conformation Stabilization. Chemistry, 26, 2020
创建时间:
2019-11-26



