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The 2.6 A Crystal Structure of a Human A2A Adenosine Receptor bound to ZM241385.

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Protein Data Bank Japan2024-10-30 更新2026-03-21 收录
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The 2.6 A Crystal Structure of a Human A2A Adenosine Receptor bound to ZM241385. Descriptor: 4-{2-[(7-amino-2-furan-2-yl[1,2,4]triazolo[1,5-a][1,3,5]triazin-5-yl)amino]ethyl}phenol, Human Adenosine A2A receptor/T4 lysozyme chimera, STEARIC ACID, ... Authors: Jaakola, V.-P, Griffith, M.T, Hanson, M.A, Cherezov, V, Chien, E.Y.T, Lane, J.R, Ijzerman, A.P, Stevens, R.C, Accelerated Technologies Center for Gene to 3D Structure (ATCG3D), GPCR Network (GPCR) Deposit date: 2008-09-24 Release date: 2008-10-14 Last modified: 2024-10-30 Method: X-RAY DIFFRACTION (2.6 Å) Cite: The 2.6 Angstrom Crystal Structure of a Human A2A Adenosine Receptor Bound to an Antagonist. Science, 322, 2008
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2008-09-24
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