five

PIM1 kinase in complex with Cpd1 (1-methyl-4-(3-(6-(piperazin-1-yl)pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl)piperazin-2-one)

收藏
Protein Data Bank Japan2024-03-06 更新2026-03-21 收录
下载链接:
https://pdbj.org/mine/summary/5v80
下载链接
链接失效反馈
官方服务:
资源简介:
PIM1 kinase in complex with Cpd1 (1-methyl-4-(3-(6-(piperazin-1-yl)pyridin-2-yl)-1H-pyrazolo[3,4-c]pyridin-5-yl)piperazin-2-one) Descriptor: 1-methyl-4-{3-[6-(piperazin-1-yl)pyridin-2-yl]-1H-pyrazolo[3,4-c]pyridin-5-yl}piperazin-2-one, PHOSPHATE ION, Serine/threonine-protein kinase pim-1 Authors: Murray, J.M, Wallweber, H. Deposit date: 2017-03-21 Release date: 2018-04-18 Last modified: 2024-03-06 Method: X-RAY DIFFRACTION (2.252 Å) Cite: Discovery of 5-Azaindazole (GNE-955) as a Potent Pan-Pim Inhibitor with Optimized Bioavailability. J. Med. Chem., 60, 2017
创建时间:
2017-03-21
二维码
社区交流群
二维码
科研交流群
商业服务