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CRYSTAL STRUCTURE OF ABL KINASE DOMAIN IN COMPLEX WITH A SMALL MOLECULE INHIBITOR

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Protein Data Bank Japan2024-03-13 更新2026-03-21 收录
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CRYSTAL STRUCTURE OF ABL KINASE DOMAIN IN COMPLEX WITH A SMALL MOLECULE INHIBITOR Descriptor: N-[4-METHYL-3-[[4-(3-PYRIDINYL)-2-PYRIMIDINYL]AMINO]PHENYL]-3-PYRIDINECARBOXAMIDE, PROTO-ONCOGENE TYROSINE-PROTEIN KINASE ABL Authors: Schindler, T, Bornmann, W, Pellicena, P, Miller, W.T, Clarkson, B, Kuriyan, J. Deposit date: 2000-08-31 Release date: 2000-09-20 Last modified: 2024-03-13 Method: X-RAY DIFFRACTION (2.4 Å) Cite: Structural mechanism for STI-571 inhibition of abelson tyrosine kinase. Science, 289, 2000
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2000-08-31
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