Src M314L T338M double mutant bound to kinase inhibitor bosutinib
收藏Protein Data Bank Japan2024-02-28 更新2026-03-21 收录
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Src M314L T338M double mutant bound to kinase inhibitor bosutinib Descriptor: 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile, Proto-oncogene tyrosine-protein kinase Src Authors: Levinson, N.M, Boxer, S.G. Deposit date: 2013-09-26 Release date: 2013-12-04 Last modified: 2024-02-28 Method: X-RAY DIFFRACTION (2.582 Å) Cite: A conserved water-mediated hydrogen bond network defines bosutinib's kinase selectivity. Nat.Chem.Biol., 10, 2014
创建时间:
2013-09-26



