five

The Fk1-Fk2 domains of FKBP52 in complex with iFit-FL

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Protein Data Bank Japan2023-12-20 更新2026-03-21 收录
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The Fk1-Fk2 domains of FKBP52 in complex with iFit-FL Descriptor: 2-(5-{[({3-[(1R)-1-[({(2S)-1-[(2S)-2-[(1S)-cyclohex-2-en-1-yl]-2-(3,4,5-trimethoxyphenyl)acetyl]piperidin-2-yl}carbonyl)oxy]-3-(3,4-dimethoxyphenyl)propyl]phenoxy}acetyl)amino]methyl}-6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid, Peptidyl-prolyl cis-trans isomerase FKBP4 Authors: Gaali, S, Kirschner, A, Cuboni, S, Hartmann, J, Kozany, C, Balsevich, G, Namendorf, C, Fernandez-Vizarra, P, Almeida, O.F.X, Ruehter, G, Uhr, M, Schmidt, M.V, Touma, C, Bracher, A, Hausch, F. Deposit date: 2014-06-30 Release date: 2014-11-26 Last modified: 2023-12-20 Method: X-RAY DIFFRACTION (3.003 Å) Cite: Selective inhibitors of the FK506-binding protein 51 by induced fit. Nat.Chem.Biol., 11, 2015
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2014-06-30
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