Bromodomain-containing 2 BD2 in complex with the inhibitor CRCM5484
收藏Protein Data Bank Japan2024-01-31 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7q5o
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Bromodomain-containing 2 BD2 in complex with the inhibitor CRCM5484 Descriptor: 1,2-ETHANEDIOL, 2-[[11-ethanoyl-4-(furan-2-ylmethyl)-3-oxidanylidene-8-thia-4,6,11-triazatricyclo[7.4.0.0^{2,7}]trideca-1(9),2(7),5-trien-5-yl]sulfanyl]-~{N}-(2-methylpyridin-3-yl)ethanamide, Bromodomain-containing protein 2 Authors: Carrasco, K, Betzi, S, Morelli, X. Deposit date: 2021-11-04 Release date: 2022-04-20 Last modified: 2024-01-31 Method: X-RAY DIFFRACTION (1.519 Å) Cite: CRCM5484: A BET-BDII Selective Compound with Differential Anti-leukemic Drug Modulation J.Med.Chem., 65, 2022
创建时间:
2021-11-04



