LSD1-CoREST1 in complex with quinazoline-derivative reversible inhibitor
收藏Protein Data Bank Japan2024-01-10 更新2026-03-21 收录
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LSD1-CoREST1 in complex with quinazoline-derivative reversible inhibitor Descriptor: FLAVIN-ADENINE DINUCLEOTIDE, Lysine-specific histone demethylase 1A, N~4~-(1-benzylpiperidin-4-yl)-N~2~-[3-(dimethylamino)propyl]-6,7-dimethoxyquinazoline-2,4-diamine, ... Authors: Speranzini, V, Rotili, D, Ciossani, G, Pilotto, S, Forgione, M, Lucidi, A, Forneris, F, Velankar, S, Mai, A, Mattevi, A. Deposit date: 2016-04-10 Release date: 2016-09-21 Last modified: 2024-01-10 Method: X-RAY DIFFRACTION (2.8 Å) Cite: Polymyxins and quinazolines are LSD1/KDM1A inhibitors with unusual structural features. Sci Adv, 2, 2016
创建时间:
2016-04-10



