Triazole-based BET family bromodomain inhibitor bound to BRD4(D1)
收藏Protein Data Bank Japan2023-10-18 更新2026-03-21 收录
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Triazole-based BET family bromodomain inhibitor bound to BRD4(D1) Descriptor: 4-{5-[6-(3,5-dimethylanilino)pyridin-2-yl]-4-methyl-1H-1,2,3-triazol-1-yl}piperidine-1-carboximidamide, Bromodomain-containing protein 4 Authors: Johnson, J.A, Pomerantz, W. Deposit date: 2021-03-12 Release date: 2021-09-29 Last modified: 2023-10-18 Method: X-RAY DIFFRACTION (1.42 Å) Cite: Systematically Mitigating the p38alpha Activity of Triazole-based BET Inhibitors ACS Med. Chem. Lett., 10, 2019
创建时间:
2021-03-12



