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Crystal Structure of Mycobacterium tuberculosis Proteasome in Complex with Phenylimidazole-based Inhibitor B6

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Protein Data Bank Japan2023-10-11 更新2026-03-21 收录
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Crystal Structure of Mycobacterium tuberculosis Proteasome in Complex with Phenylimidazole-based Inhibitor B6 Descriptor: N-{(2S)-1-({(1S)-1-[5-(2-fluorophenyl)-1H-imidazol-2-yl]ethyl}amino)-1,4-dioxo-4-[(2R)-2-phenylpyrrolidin-1-yl]butan-2-yl}-5-methyl-1,2-oxazole-3-carboxamide, Proteasome subunit alpha, Proteasome subunit beta Authors: Hsu, H.C, Li, H. Deposit date: 2019-03-26 Release date: 2019-10-09 Last modified: 2023-10-11 Method: X-RAY DIFFRACTION (2.9 Å) Cite: Selective Phenylimidazole-Based Inhibitors of theMycobacterium tuberculosisProteasome. J.Med.Chem., 62, 2019
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2019-03-26
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