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ERAP1 in complex with 1-[2-(3-oxo-6-phenyl-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamido]cyclohexane-1-carboxylic acid

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Protein Data Bank Japan2026-05-06 更新2026-08-24 收录
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ERAP1 in complex with 1-[2-(3-oxo-6-phenyl-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamido]cyclohexane-1-carboxylic acid Descriptor: 1,2-ETHANEDIOL, 1-[2-(3-oxidanylidene-6-phenyl-1,4-benzoxazin-4-yl)ethanoylamino]cyclohexane-1-carboxylic acid, Endoplasmic reticulum aminopeptidase 1, ... Authors: Rowland, P. Deposit date: 2025-11-22 Release date: 2026-04-22 Last modified: 2026-05-06 Method: X-RAY DIFFRACTION (1.37 Å) Cite: Automated Molecular Design in BRADSHAW, Applied to the Optimization of ERAP1 Inhibitors. J.Med.Chem., 69, 2026

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2025-11-22
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