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X-ray structure of human PPAR delta ligand binding domain-pemafibrate co-crystals obtained by co-crystallization

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Protein Data Bank Japan2023-11-29 更新2026-04-19 收录
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https://pdbj.org/mine/summary/7wgn
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X-ray structure of human PPAR delta ligand binding domain-pemafibrate co-crystals obtained by co-crystallization Descriptor: (2~{R})-2-[3-[[1,3-benzoxazol-2-yl-[3-(4-methoxyphenoxy)propyl]amino]methyl]phenoxy]butanoic acid, Peroxisome proliferator-activated receptor delta, octyl beta-D-glucopyranoside Authors: Kamata, S, Honda, A, Akahane, M, Machida, Y, Uchii, K, Shiiyama, Y, Masuda, R, Oyama, T, Ishii, I. Deposit date: 2021-12-28 Release date: 2022-05-25 Last modified: 2023-11-29 Method: X-RAY DIFFRACTION (1.813 Å) Cite: Functional and Structural Insights into Human PPAR alpha / delta / gamma Subtype Selectivity of Bezafibrate, Fenofibric Acid, and Pemafibrate. Int J Mol Sci, 23, 2022
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2021-12-28
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