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Crystal structure of SARS-Cov-2 main protease G15S mutant in complex with Bofutrelvir

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Protein Data Bank Japan2025-04-09 更新2026-04-04 收录
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Crystal structure of SARS-Cov-2 main protease G15S mutant in complex with Bofutrelvir Descriptor: 3C-like proteinase nsp5, ~{N}-[(2~{S})-3-cyclohexyl-1-oxidanylidene-1-[[(2~{S})-1-oxidanylidene-3-[(3~{S})-2-oxidanylidenepyrrolidin-3-yl]propan-2-yl]amino]propan-2-yl]-1~{H}-indole-2-carboxamide Authors: Zeng, P, Wang, W.W, Zhang, J, Li, J. Deposit date: 2024-01-30 Release date: 2025-01-08 Last modified: 2025-04-09 Method: X-RAY DIFFRACTION (1.93 Å) Cite: Inhibitory efficacy and structural insights of Bofutrelvir against SARS-CoV-2 M pro mutants and MERS-CoV M pro. Commun Biol, 8, 2025
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2024-01-30
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