five

TTK kinase domain in complex with a PEG-linked pyrimido-indolizine

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Protein Data Bank Japan2024-10-16 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5na0
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TTK kinase domain in complex with a PEG-linked pyrimido-indolizine Descriptor: Dual specificity protein kinase TTK, ~{N}-[3,5-diethyl-1-[2-[2-(2-methoxyethoxy)ethoxy]ethyl]pyrazol-4-yl]-2-[[2-methoxy-4-[4-(2-methoxyethanoyl)piperazin-1-yl]phenyl]amino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamide Authors: Uitdehaag, J, Willemsen-Seegers, N, de Man, J, Buijsman, R.C, Zaman, G.J.R. Deposit date: 2017-02-27 Release date: 2017-05-31 Last modified: 2024-10-16 Method: X-RAY DIFFRACTION (2.9 Å) Cite: Target Residence Time-Guided Optimization on TTK Kinase Results in Inhibitors with Potent Anti-Proliferative Activity. J. Mol. Biol., 429, 2017
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2017-02-27
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