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KRAS G12C in bound to quinazoline based switch II pocket (SWIIP) binder

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Protein Data Bank Japan2024-11-06 更新2026-03-21 收录
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https://pdbj.org/mine/summary/5v71
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KRAS G12C in bound to quinazoline based switch II pocket (SWIIP) binder Descriptor: 1-{4-[6-chloro-7-(2-fluorophenyl)quinazolin-4-yl]piperazin-1-yl}propan-1-one, GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, ... Authors: Westover, K, Lu, J. Deposit date: 2017-03-17 Release date: 2017-08-23 Last modified: 2024-11-06 Method: X-RAY DIFFRACTION (2.228 Å) Cite: KRAS G12C Drug Development: Discrimination between Switch II Pocket Configurations Using Hydrogen/Deuterium-Exchange Mass Spectrometry. Structure, 25, 2017
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2017-03-17
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